Publications

  • Mitran, Bogdan; Varasteh, Zohreh; Puuvuori, Emmi; Abousayed, Ayman et al.

    Bispecific GRPR-antagonistic anti-PSMA/GRPR heterodimer for PET and SPECT diagnostic imaging of prostate cancer

    Part of Cancers, 2019.

  • Shariatgorji, Mohammadreza; Nilsson, Anna; Fridjonsdottir, Elva; Vallianatou, Theodosia et al.

    Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

    Part of Nature Methods, p. 1021-1028, 2019.

  • Oroujeni, Maryam; Abouzayed, Ayman; Lundmark, Fanny; Mitran, Bogdan et al.

    Evaluation of Tumor-Targeting Properties of an Antagonistic Bombesin Analogue RM26 Conjugated with a Non-Residualizing Radioiodine Label Comparison with a Radiometal-Labelled Counterpart

    Part of Pharmaceutics, 2019.

    Open access
  • Abouzayed, Ayman; Yim, Cheng-Bin; Mitran, Bogdan; Rinne, Sara S. et al.

    Synthesis and Preclinical Evaluation of Radio-Iodinated GRPR/PSMA Bispecific Heterodimers for the Theranostics Application in Prostate Cancer

    Part of Pharmaceutics, 2019.

    Open access
  • Schembri, Luke S; Eriksson, Jonas; Odell, Luke R.

    Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

    Part of Journal of Organic Chemistry, p. 6970-6981, 2019.

  • Mitran, Bogdan; Rinne, Sara S.; Konijnenberg, Mark W.; Maina, Theodosia et al.

    Trastuzumab cotreatment improves survival of mice with PC-3 prostate cancer xenografts treated with the GRPR antagonist 177Lu-DOTAGA-PEG2-RM26

    Part of International Journal of Cancer, p. 3347-3358, 2019.

    Open access
  • Söderström, Marcus; Zamaratski, Edouard; Odell, Luke R.

    Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF3⦁SMe2

    Part of European Journal of Organic Chemistry, p. 5402-5408, 2019.

    Open access
  • Eriksson, Jonas; Roy, Tamal; Sawadjoon, Supaporn; Bachmann, Kim et al.

    Synthesis and preclinical evaluation of the CRTH2 antagonist [11C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

    Part of Nuclear Medicine and Biology, p. 1-10, 2019.

    Open access
  • Isaksson, Rebecka; Lindman, Jens; Wannberg, Johan; Sallander, Jessica et al.

    A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode

    Part of ChemistryOpen, p. 114-125, 2019.

    Open access
  • Åkerbladh, Linda; Odell, Luke R.; Larhed, Mats

    Palladium-Catalyzed Molybdenum Hexacarbonyl-Mediated Gas-Free Carbonylative Reactions

    Part of Synlett, p. 141-155, 2019.

  • Adeyemi, Ahmed; Wetzel, Alexander; Bergman, Joakim; Brånalt, Jonas et al.

    Regio- and Stereoselective Synthesis of Spirooxindoles via Mizoroki-Heck Coupling of Aryl Iodides

    Part of Synlett, p. 82-88, 2019.

  • Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

    Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones

    Part of ACS OMEGA, p. 14258 14258-14265 14265, 2018.

    Open access
  • Reddy Vanga, Sudarsana; Sävmarker, Jonas; Ng, Leelee; Larhed, Mats et al.

    Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides

    Part of ACS OMEGA, p. 4509 4509-4521 4521, 2018.

    Open access
  • Wannberg, Johan; Isaksson, Rebecka; Bremberg, Ulf; Backlund, Maria et al.

    A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes

    Part of Bioorganic & Medicinal Chemistry Letters, p. 519-522, 2018.

  • Monazzam, Azita; Lau, Joey; Velikyan, Irina; Li, Su-Chen et al.

    Increased Expression of GLP-1R in Proliferating Islets of Men1 Mice is Detectable by [Ga-68]Ga-DO3A-VS-Cys(40)- Exendin-4/PET

    Part of Scientific Reports, 2018.

    Open access
  • Chow, Shiao Y.; Odell, Luke R.; Eriksson, Jonas

    Low-Pressure Radical 11C-Aminocarbonylation of Alkyl Iodides through Thermal Initiation

    Part of European Journal of Organic Chemistry, p. 1236-1236, 2017.

  • Åkerbladh, Linda; Schembri, Luke S; Larhed, Mats; Odell, Luke R.

    Palladium(0)-Catalyzed Carbonylative One-Pot Synthesis of N-Acylguanidines

    Part of Journal of Organic Chemistry, p. 12520-12529, 2017.

  • Eriksson, Olof; Rosenström, Ulrika; Selvaraju, Ram Kumar; Eriksson, Barbro et al.

    Species differences in pancreatic binding of DO3A-VS-Cys40-Exendin4

    Part of Acta Diabetologica, p. 1039-1045, 2017.

    Open access
  • Kumaniaev, Ivan; Subbotina, Elena; Sävmarker, Jonas; Larhed, Mats et al.

    Lignin depolymerization to monophenolic compounds in a flow-through system

    Part of Green Chemistry, p. 5767-5771, 2017.

  • Velikyan, Irina; Rosenström, Ulrika; Eriksson, Olof

    Fully automated GMP production of [Ga-68]Ga-DO3A-VS-Cys(40)-Exendin-4 for clinical use

    Part of American Journal of Nuclear Medicine and Molecular Imaging, p. 111-125, 2017.

    Open access
  • Mitran, Bogdan; Thisgaard, Helge; Rosenström, Ulrika; Dam, Johan Hygum et al.

    High Contrast PET Imaging of GRPR Expression in Prostate Cancer Using Cobalt-Labeled Bombesin Antagonist RM26

    Part of Contrast Media & Molecular Imaging, 2017.

    Open access
  • Adeyemi, Ahmed; Bergman, Joakim; Branalt, Jonas; Sävmarker, Jonas et al.

    Continuous Flow Synthesis under High-Temperature/High-Pressure Conditions Using a Resistively Heated Flow Reactor

    Part of Organic Process Research & Development, p. 947-955, 2017.

  • Bergman, Sara; Brandt, Peter; Nordeman, Patrik; Larhed, Mats et al.

    Synthesis of 11C-Labelled Ureas by Palladium(II)-Mediated Oxidative Carbonylation

    Part of Molecules, 2017.

    Open access
  • Roslin, Sara; De Rosa, Maria; Deuther-Conrad, Winnie; Eriksson, Jonas et al.

    Synthesis and In Vitro Evaluation of 5-Substituted Benzovesamicol Analogs containing N-Substituted Amides as Potential Positron Emission Tomography Tracers for the Vesicular Acetylcholine Transporter

    Part of Bioorganic & Medicinal Chemistry, p. 5095-5106, 2017.

  • Roslin, Sara; Odell, Luke R.

    Palladium and Visible-Light Mediated Carbonylative Suzuki-Miyaura Coupling of Unactivated Alkyl Halides and Aryl Boronic Acids

    Part of Chemical Communications, p. 6895-6898, 2017.

  • Åkerbladh, Linda; Chow, Shiao Y.; Odell, Luke R.; Larhed, Mats

    Synthesis of 4H-Benzo[e][1,3]oxazin-4-ones by a Carbonylation-Cyclization Domino Reaction of ortho-Halophenols and Cyanamide

    Part of ChemistryOpen, p. 620-628, 2017.

    Open access
  • Nordeman, Patrik; Chow, Shiao Y.; Odell, A. F.; Antoni, Gunnar et al.

    Palladium-mediated C-11-carbonylations using aryl halides and cyanamide

    Part of Organic and biomolecular chemistry, p. 4875-4881, 2017.

  • Roy, Tamal; Brandt, Peter; Wetzel, Alexander; Bergman, Joakim et al.

    Selective Synthesis of Spirooxindoles by an Intramolecular Heck-Mizoroki Reaction

    Part of Organic Letters, p. 2738-2741, 2017.

  • Rydfjord, Jonas; Skillinghaug, Bobo; Brandt, Peter; Odell, Luke R. et al.

    Route to 3-Amidino Indoles via Pd(II)-Catalyzed C-H Bond Activation

    Part of Organic Letters, p. 4066-4069, 2017.

  • Roslin, Sara; Odell, Luke R.

    Visible-Light Photocatalysis as an Enabling Tool for the Functionalization of Unactivated C(sp(3))-Substrates

    Part of European Journal of Organic Chemistry, p. 1993-2007, 2017.

  • Chow, Shiao Y.; Odell, Luke R.

    Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

    Part of Journal of Organic Chemistry, p. 2515-2522, 2017.

  • Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

    Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

    Part of Chemical Communications, p. 2110-2113, 2017.

  • Wetzel, Alexander; Bergman, Joakim; Brandt, Peter; Larhed, Mats et al.

    Regio- and Stereoselective Synthesis of Functionalized Cyclopentene Derivatives via Mizoroki-Heck Reactions.

    Part of Organic Letters, p. 1602-1605, 2017.

  • Odell, Luke R.; Abdel-Hamid, Mohammed K.; Hill, Timothy A.; Chau, Ngoc et al.

    Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain

    Part of Journal of Medicinal Chemistry, p. 349-361, 2017.

  • Stevens, Marc Y.; Chow, Shiao Y.; Estrada, Sergio; Eriksson, Jonas et al.

    Synthesis of C-11-labeled Sulfonyl Carbamates through a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols, and [C-11]CO

    Part of ChemistryOpen, p. 566-573, 2016.

    Open access
  • Chow, Shiao Y.; Odell, Luke R.; Eriksson, Jonas

    Low-Pressure Radical C-11-Aminocarbonylation of Alkyl Iodides through Thermal Initiation

    Part of European Journal of Organic Chemistry, p. 5980-5989, 2016.

  • Velikyan, Irina; Rosenström, Ulrika; Eriksson, Olof; Antoni, Gunnar

    Ga-68/PET imaging and quantification of fibrosis using peptide-based tracers

    Part of European Journal of Nuclear Medicine and Molecular Imaging, p. S73-S73, 2016.

  • Sawant, Rajiv T.; Stevens, Marc Y.; Sköld, Christian; Odell, Luke R.

    Microwave-Assisted Branching Cascades: A Route to Diverse 3,4-Dihydroquinazolinone-Embedded Polyheterocyclic Scaffolds

    Part of Organic Letters, p. 5392-5395, 2016.

  • Diwakarla, Shanti; Nylander, Erik; Grönbladh, Alfhild; Vanga, Sudarsana Reddy et al.

    Aryl Sulfonamide Inhibitors of Insulin-Regulated Aminopeptidase Enhance Spine Density in Primary Hippocampal Neuron Cultures

    Part of ACS Chemical Neuroscience, p. 1383-1392, 2016.

  • Skillinghaug, Bobo; Rydfjord, Jonas; Sävmarker, Jonas; Larhed, Mats

    Microwave Heated Continuous Flow Palladium(II)-Catalyzed Desulfitative Synthesis of Aryl Ketones

    Part of Organic Process Research & Development, p. 2005-2011, 2016.

  • Chow, Shiao Y.; Stevens, Marc Y.; Åkerbladh, Linda; Bergman, Sara et al.

    Mild and Low-Pressure fac-Ir(ppy)3-Mediated Radical Aminocarbonylation of Unactivated Alkyl Iodides through Visible-Light Photoredox Catalysis

    Part of Chemistry - A European Journal, p. 9155-9161, 2016.

  • Engen, Karin; Rosenström, Ulrika; Axelsson, Hanna; Konda, Vivek et al.

    Identification of Drug-Like Inhibitors of Insulin-Regulated Aminopeptidase Through Small-Molecule Screening

    Part of Assay and drug development technologies, p. 180-193, 2016.

  • Stevens, Marc; Chow, Chow; Estrada, Sergio; Eriksson, Jonas et al.

    Synthesis of 11C-labelled Sulfonyl Carbamates via a Multicomponent Reaction Employing Sulfonyl Azides, Alcohols and [11C]CO

    Part of ChemistryOpen, p. 566-573, 2016.

  • Åkerbladh, Linda; Odell, Luke R.

    Synthesis of 2-Aminoquinazolinones via Carbonylative Coupling of ortho-lodoanilines and Cyanamide

    Part of Journal of Organic Chemistry, p. 2966-2973, 2016.

  • Isaksson, Rebecka; Kumpina, Ilze; Larhed, Mats; Wannberg, Johan

    Rapid and straightforward transesterification of sulfonyl carbamates

    Part of Tetrahedron Letters, p. 1476-1478, 2016.

  • Kumpina, Ilze; Isaksson, Rebecka; Sävmarker, Jonas; Wannberg, Johan et al.

    Microwave Promoted Transcarbamylation Reaction of Sulfonylcarbamates under Continuous-Flow Conditions

    Part of Organic Process Research & Development, p. 440-445, 2016.

  • Mitran, Bogdan; Varasteh, Zohreh; Selvaraju, Ram Kumar; Lindeberg, Gunnar et al.

    Selection of optimal chelator improves the contrast of GRPR imaging using bombesin analogue RM26.

    Part of International journal of oncology, p. 2124-2134, 2016.

  • Chow, Shiao; Stevens, Marc; Odell, Luke

    Sulfonyl Azides as Precursors in Ligand-free Palladium-Catalyzed Synthesis of Sulfonyl Carbamates and Sulfonyl Ureas and Synthesis of Sulfonamides

    Part of Journal of Organic Chemistry, p. 2681-2691, 2016.

  • Skillinghaug, Bobo; Rydfjord, Jonas; Odell, Luke R.

    Synthesis of sodium aryl sulfinates from aryl bromides employing 1,4-diazabicyclo[2.2.2]octane bis(sulfur dioxide) adduct (DABSO) as a bench-stable, gas-free alternative to SO2

    Part of Tetrahedron Letters, p. 533-536, 2016.

  • Diwakarla, Shanti; Nylander, Erik; Grönbladh, Alfhild; Reddy Vanga, Sudarsana et al.

    Binding to and Inhibition of Insulin-Regulated Aminopeptidase (IRAP) by Macrocyclic Disulfides Enhances Spine Density

    Part of Molecular Pharmacology, p. 413-424, 2016.