Publikationer

  • Åkerbladh, Linda; Odell, Luke R.; Larhed, Mats

    Palladium-Catalyzed Molybdenum Hexacarbonyl-Mediated Gas-Free Carbonylative Reactions

    Ingår i Synlett, s. 141-155, 2019.

  • Adeyemi, Ahmed; Wetzel, Alexander; Bergman, Joakim; Brånalt, Jonas et al.

    Regio- and Stereoselective Synthesis of Spirooxindoles via Mizoroki-Heck Coupling of Aryl Iodides

    Ingår i Synlett, s. 82-88, 2019.

  • Isaksson, Rebecka; Lindman, Jens; Wannberg, Johan; Sallander, Jessica et al.

    A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode

    Ingår i ChemistryOpen, s. 114-125, 2019.

    Open access
  • Schembri, Luke S; Eriksson, Jonas; Odell, Luke R.

    Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

    Ingår i Journal of Organic Chemistry, s. 6970-6981, 2019.

  • Mitran, Bogdan; Rinne, Sara S.; Konijnenberg, Mark W.; Maina, Theodosia et al.

    Trastuzumab cotreatment improves survival of mice with PC-3 prostate cancer xenografts treated with the GRPR antagonist 177Lu-DOTAGA-PEG2-RM26

    Ingår i International Journal of Cancer, 2019.

    Open access
  • Eriksson, Jonas; Roy, Tamal; Sawadjoon, Supaporn; Bachmann, Kim et al.

    Synthesis and preclinical evaluation of the CRTH2 antagonist [11C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

    Ingår i Nuclear Medicine and Biology, s. 1-10, 2019.

    Open access
  • Abouzayed, Ayman; Yim, Cheng-Bin; Mitran, Bogdan; Rinne, Sara S. et al.

    Synthesis and Preclinical Evaluation of Radio-Iodinated GRPR/PSMA Bispecific Heterodimers for the Theranostics Application in Prostate Cancer

    Ingår i Pharmaceutics, 2019.

    Open access
  • Oroujeni, Maryam; Abouzayed, Ayman; Lundmark, Fanny; Mitran, Bogdan et al.

    Evaluation of Tumor-Targeting Properties of an Antagonistic Bombesin Analogue RM26 Conjugated with a Non-Residualizing Radioiodine Label Comparison with a Radiometal-Labelled Counterpart

    Ingår i Pharmaceutics, 2019.

    Open access
  • Monazzam, Azita; Lau, Joey; Velikyan, Irina; Li, Su-Chen et al.

    Increased Expression of GLP-1R in Proliferating Islets of Men1 Mice is Detectable by [Ga-68]Ga-DO3A-VS-Cys(40)- Exendin-4/PET

    Ingår i Scientific Reports, 2018.

    Open access
  • Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

    Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones

    Ingår i ACS OMEGA, s. 14258 14258-14265 14265, 2018.

    Open access
  • Wannberg, Johan; Isaksson, Rebecka; Bremberg, Ulf; Backlund, Maria et al.

    A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes

    Ingår i Bioorganic & Medicinal Chemistry Letters, s. 519-522, 2018.

  • Reddy Vanga, Sudarsana; Sävmarker, Jonas; Ng, Leelee; Larhed, Mats et al.

    Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides

    Ingår i ACS OMEGA, s. 4509 4509-4521 4521, 2018.

    Open access
  • Roslin, Sara; Odell, Luke R.

    Palladium and Visible-Light Mediated Carbonylative Suzuki-Miyaura Coupling of Unactivated Alkyl Halides and Aryl Boronic Acids

    Ingår i Chemical Communications, s. 6895-6898, 2017.

  • Adeyemi, Ahmed; Bergman, Joakim; Branalt, Jonas; Sävmarker, Jonas et al.

    Continuous Flow Synthesis under High-Temperature/High-Pressure Conditions Using a Resistively Heated Flow Reactor

    Ingår i Organic Process Research & Development, s. 947-955, 2017.

  • Roy, Tamal; Brandt, Peter; Wetzel, Alexander; Bergman, Joakim et al.

    Selective Synthesis of Spirooxindoles by an Intramolecular Heck-Mizoroki Reaction

    Ingår i Organic Letters, s. 2738-2741, 2017.

  • Roslin, Sara; Odell, Luke R.

    Visible-Light Photocatalysis as an Enabling Tool for the Functionalization of Unactivated C(sp(3))-Substrates

    Ingår i European Journal of Organic Chemistry, s. 1993-2007, 2017.

  • Velikyan, Irina; Rosenström, Ulrika; Eriksson, Olof

    Fully automated GMP production of [Ga-68]Ga-DO3A-VS-Cys(40)-Exendin-4 for clinical use

    Ingår i American Journal of Nuclear Medicine and Molecular Imaging, s. 111-125, 2017.

    Open access
  • Chow, Shiao Y.; Odell, Luke R.

    Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

    Ingår i Journal of Organic Chemistry, s. 2515-2522, 2017.

  • Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

    Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

    Ingår i Chemical Communications, s. 2110-2113, 2017.

  • Wetzel, Alexander; Bergman, Joakim; Brandt, Peter; Larhed, Mats et al.

    Regio- and Stereoselective Synthesis of Functionalized Cyclopentene Derivatives via Mizoroki-Heck Reactions.

    Ingår i Organic Letters, s. 1602-1605, 2017.

  • Odell, Luke R.; Abdel-Hamid, Mohammed K.; Hill, Timothy A.; Chau, Ngoc et al.

    Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain

    Ingår i Journal of Medicinal Chemistry, s. 349-361, 2017.

  • Nordeman, Patrik; Chow, Shiao Y.; Odell, A. F.; Antoni, Gunnar et al.

    Palladium-mediated C-11-carbonylations using aryl halides and cyanamide

    Ingår i Organic and biomolecular chemistry, s. 4875-4881, 2017.

  • Rydfjord, Jonas; Skillinghaug, Bobo; Brandt, Peter; Odell, Luke R. et al.

    Route to 3-Amidino Indoles via Pd(II)-Catalyzed C-H Bond Activation

    Ingår i Organic Letters, s. 4066-4069, 2017.

  • Åkerbladh, Linda; Chow, Shiao Y.; Odell, Luke R.; Larhed, Mats

    Synthesis of 4H-Benzo[e][1,3]oxazin-4-ones by a Carbonylation-Cyclization Domino Reaction of ortho-Halophenols and Cyanamide

    Ingår i ChemistryOpen, s. 620-628, 2017.

    Open access
  • Kumaniaev, Ivan; Subbotina, Elena; Sävmarker, Jonas; Larhed, Mats et al.

    Lignin depolymerization to monophenolic compounds in a flow-through system

    Ingår i Green Chemistry, s. 5767-5771, 2017.

  • Eriksson, Olof; Rosenström, Ulrika; Selvaraju, Ram Kumar; Eriksson, Barbro et al.

    Species differences in pancreatic binding of DO3A-VS-Cys40-Exendin4

    Ingår i Acta Diabetologica, s. 1039-1045, 2017.

    Open access
  • Chow, Shiao Y.; Odell, Luke R.; Eriksson, Jonas

    Low-Pressure Radical 11C-Aminocarbonylation of Alkyl Iodides through Thermal Initiation

    Ingår i European Journal of Organic Chemistry, s. 1236-1236, 2017.

  • Åkerbladh, Linda; Schembri, Luke S; Larhed, Mats; Odell, Luke R.

    Palladium(0)-Catalyzed Carbonylative One-Pot Synthesis of N-Acylguanidines

    Ingår i Journal of Organic Chemistry, s. 12520-12529, 2017.

  • Bergman, Sara; Brandt, Peter; Nordeman, Patrik; Larhed, Mats et al.

    Synthesis of 11C-Labelled Ureas by Palladium(II)-Mediated Oxidative Carbonylation

    Ingår i Molecules, 2017.

    Open access
  • Roslin, Sara; De Rosa, Maria; Deuther-Conrad, Winnie; Eriksson, Jonas et al.

    Synthesis and In Vitro Evaluation of 5-Substituted Benzovesamicol Analogs containing N-Substituted Amides as Potential Positron Emission Tomography Tracers for the Vesicular Acetylcholine Transporter

    Ingår i Bioorganic & Medicinal Chemistry, s. 5095-5106, 2017.