Publikationer

  • Nordeman, Patrik; Jayendra, Z. P.; Briard, E.; Li, Su-Chen et al.

    18F-Radiolabeling and Preliminary Evaluation of a HSP90 ligand

    Ingår i European Journal of Pharmaceutical Sciences, 2021.

  • Fridjonsdottir, Elva; Shariatgorji, Mohammadreza; Nilsson, Anna; Vallianatou, Theodosia et al.

    Mass spectrometry imaging identifies abnormally elevated brain L-DOPA levels and extrastriatal monoaminergic dysregulation in L-DOPA-induced dyskinesia

    Ingår i Science Advances, 2021.

    Open access
  • Wannberg, Johan; Gising, Johan; Lindman, Jens; Salander, Jessica et al.

    N-(Methyloxycarbonyl)thiophene sulfonamides as high affinity AT2 receptor ligands

    Ingår i Bioorganic & Medicinal Chemistry, 2021.

  • Rosestedt, Maria; Velikyan, Irina; Rosenström, Ulrika; Estrada, Sergio et al.

    Radiolabelling and positron emission tomography imaging of a high-affinity peptide binder to collagen type 1

    Ingår i Nuclear Medicine and Biology, s. 54-62, 2021.

    Open access
  • Bokale-Shivale, Suvarna; Amin, Mohammad A.; Sawant, Rajiv T.; Stevens, Marc Y. et al.

    Synthesis of substituted 3,4-dihydroquinazolinones via a metal free Leuckart-Wallach type reaction

    Ingår i RSC Advances, s. 349-353, 2021.

    Open access
  • Cheung, Pierre; Zhang, Bo; Puuvuori, Emmi; Estrada, Sergio et al.

    PET Imaging of GPR44 by Antagonist [C-11]MK-7246 in Pigs

    Ingår i BIOMEDICINES, 2021.

    Open access
  • Isaksson, Rebecka; Casselbrant, Anna; Elebring, Erik; Hallberg, Mathias et al.

    Direct stimulation of angiotensin II type 2 receptor reduces nitric oxide production in lipopolysaccharide treated mouse macrophages

    Ingår i European Journal of Pharmacology, 2020.

    Open access
  • Engen, Karin; Reddy Vanga, Sudarsana; Lundbäck, Thomas; Agalo, Faith et al.

    Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors

    Ingår i ChemistryOpen, s. 325-337, 2020.

    Open access
  • Barlow, Nicholas; Reddy Vanga, Sudarsana; Sävmarker, Jonas; Sandström, Anja et al.

    Macrocyclic Peptidomimetics as Inhibitors of Insulin-Regulated Aminopeptidase (IRAP)

    Ingår i RSC Medicinal chemistry, s. 234-244, 2020.

  • Mpakali, Anastasia; Saridakis, Emmanuel; Giastas, Petros; Maben, Zachary et al.

    Structural Basis of Inhibition of Insulin-Regulated Aminopeptidase by a Macrocyclic Peptidic Inhibitor

    Ingår i ACS Medicinal Chemistry Letters, s. 1429-1434, 2020.

  • Adeyemi, Ahmed; Odell, Luke R.; Larhed, Mats

    Regio- and Stereoselective Synthesis of Allylic Spiroethers (Spirobenzofuranes) via an Intramolecular Mizoroki-Heck Reaction

    Ingår i Journal of Organic Chemistry, s. 7648-7657, 2020.

    Open access
  • Lundmark, Fanny; Abouzayed, Ayman; Mitran, Bogdan; Rinne, Sara S. et al.

    Heterodimeric Radiotracer Targeting PSMA and GRPR for Imaging of Prostate Cancer-Optimization of the Affinity towards PSMA by Linker Modification in Murine Model

    Ingår i Pharmaceutics, 2020.

    Open access
  • Ye, Sofie; Hartmann, Rafael; Söderström, Marcus; Amin, Mohammad A. et al.

    Turning Information Dissipation into Dissemination: Instagram as a Communication Enhancing Tool during the COVID-19 Pandemic and Beyond

    Ingår i Journal of Chemical Education, s. 3217-3222, 2020.

  • Hallberg, Mathias; Larhed, Mats

    From Angiotensin IV to Small Peptidemimetics Inhibiting Insulin-Regulated Aminopeptidase

    Ingår i Frontiers in Pharmacology, 2020.

    Open access
  • Hartmann, Rafael; Fahrner, Raphael; Shevshenko, Denys; Fryknäs, Mårten et al.

    Rational Design of Azastatin as a Potential ADC Payload with Reduced Bystander Killing.

    Ingår i ChemMedChem, s. 2500-2512, 2020.

    Open access
  • Isaksson, Rebecka; Lindman, Jens; Wannberg, Johan; Sallander, Jessica et al.

    A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode

    Ingår i ChemistryOpen, s. 114-125, 2019.

    Open access
  • Schembri, Luke S; Eriksson, Jonas; Odell, Luke R.

    Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

    Ingår i Journal of Organic Chemistry, s. 6970-6981, 2019.

  • Eriksson, Jonas; Roy, Tamal; Sawadjoon, Supaporn; Bachmann, Kim et al.

    Synthesis and preclinical evaluation of the CRTH2 antagonist [11C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

    Ingår i Nuclear Medicine and Biology, s. 1-10, 2019.

    Open access
  • Abouzayed, Ayman; Yim, Cheng-Bin; Mitran, Bogdan; Rinne, Sara S. et al.

    Synthesis and Preclinical Evaluation of Radio-Iodinated GRPR/PSMA Bispecific Heterodimers for the Theranostics Application in Prostate Cancer

    Ingår i Pharmaceutics, 2019.

    Open access
  • Oroujeni, Maryam; Abouzayed, Ayman; Lundmark, Fanny; Mitran, Bogdan et al.

    Evaluation of Tumor-Targeting Properties of an Antagonistic Bombesin Analogue RM26 Conjugated with a Non-Residualizing Radioiodine Label Comparison with a Radiometal-Labelled Counterpart

    Ingår i Pharmaceutics, 2019.

    Open access
  • Söderström, Marcus; Zamaratski, Edouard; Odell, Luke R.

    Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF3⦁SMe2

    Ingår i European Journal of Organic Chemistry, s. 5402-5408, 2019.

    Open access
  • Mitran, Bogdan; Rinne, Sara S.; Konijnenberg, Mark W.; Maina, Theodosia et al.

    Trastuzumab cotreatment improves survival of mice with PC-3 prostate cancer xenografts treated with the GRPR antagonist 177Lu-DOTAGA-PEG2-RM26

    Ingår i International Journal of Cancer, s. 3347-3358, 2019.

    Open access
  • Adeyemi, Ahmed; Wetzel, Alexander; Bergman, Joakim; Brånalt, Jonas et al.

    Regio- and Stereoselective Synthesis of Spirooxindoles via Mizoroki-Heck Coupling of Aryl Iodides

    Ingår i Synlett, s. 82-88, 2019.

  • Mitran, Bogdan; Varasteh, Zohreh; Abouzayed, Ayman; Rinne, Sara S. et al.

    Bispecific GRPR-antagonistic anti-PSMA/GRPR heterodimer for PET and SPECT diagnostic imaging of prostate cancer

    Ingår i Cancers, 2019.

    Open access
  • Åkerbladh, Linda; Odell, Luke R.; Larhed, Mats

    Palladium-Catalyzed Molybdenum Hexacarbonyl-Mediated Gas-Free Carbonylative Reactions

    Ingår i Synlett, s. 141-155, 2019.

  • Shariatgorji, Mohammadreza; Nilsson, Anna; Fridjonsdottir, Elva; Vallianatou, Theodosia et al.

    Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

    Ingår i Nature Methods, s. 1021-1028, 2019.

  • Mitran, Bogdan; Thisgaard, Helge; Rinne, Sara S.; Dam, Johan Hygum et al.

    Selection of an optimal macrocyclic chelator improves the imaging of prostate cancer using cobalt-labeled GRPR antagonist RM26

    Ingår i Scientific Reports, 2019.

    Open access
  • Wannberg, Johan; Isaksson, Rebecka; Bremberg, Ulf; Backlund, Maria et al.

    A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes

    Ingår i Bioorganic & Medicinal Chemistry Letters, s. 519-522, 2018.

  • Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

    Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones

    Ingår i ACS Omega, s. 14258-14265, 2018.

    Open access
  • Reddy Vanga, Sudarsana; Sävmarker, Jonas; Ng, Leelee; Larhed, Mats et al.

    Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides

    Ingår i ACS Omega, s. 4509-4521, 2018.

    Open access